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H-89(PKA抑制剂) |
产品编号: S1644
产品包装: 5mg
产品价格: 731.00元 |
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产品简介
产品简介:
H-89也称H89,全称为N-[2-(p-Bromocinnamylamino)ethyl]-5-isoquinolinesulfonamide·2HCl
hydrate,是一种常用的PKA抑制剂。H-89可以通透细胞,可以选择性抑制cAMP、cGMP依赖的蛋白激酶PKA、PKG和PKCμ,但对于PKA的选择性抑制作用更强。
H-89分子量为519.28,分子式为C20H20BrN3O2S·2HCl,CAS Number:127243-85-0。本产品为进口分
装,纯度大于98%。
H-89溶于DMSO(20mg/ml)和无水乙醇(0.15 mg/ml),难溶于水。
包装清单:
产品编号 |
产品名称 |
包装 |
S1644 |
H-89(PKA抑制剂) |
5mg |
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说明书 |
1份 |
保存条件:
-20℃保存,一年有效。
注意事项:
本产品对人体有害,操作时请小心,并注意有效防护以避免直接接触人体或吸入体内。
为了您的安全和健康,请穿实验服并戴一次性手套操作。
使用说明
使用说明:
1. 建议先使用DMSO配制成储存液后使用。H-89常见使用浓度范围为10-30μM,也有报道在1-50μM范围内使
用。具体的最佳工作浓度请参考相关文献,或根据实验目的,以及所培养的特定细胞和组织,通过实验
进行摸索和优化。
产品图片
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